SYNTHESIS OF 2'-(3-ALPHA-BENZYLOXY-24-NORCHOLAN-23-YL)-2',4',4'-TRIMETHYL-4',5'-DIHYDROOXAZOLINE-N-OXYL - A NEW POTENTIAL SPIN PROBE FOR BIOMEMBRANES
DSpace at IIT Bombay
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Title |
SYNTHESIS OF 2'-(3-ALPHA-BENZYLOXY-24-NORCHOLAN-23-YL)-2',4',4'-TRIMETHYL-4',5'-DIHYDROOXAZOLINE-N-OXYL - A NEW POTENTIAL SPIN PROBE FOR BIOMEMBRANES
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Creator |
BANERJEE, S
DESAI, UR TRIVEDI, GK |
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Subject |
labels
oxidation |
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Description |
The synthesis of a new steroidal nitroxide, viz. 2'-(3-alpha-benzyloxy-24-norcholan-23-yl)-2',4',4'-trimethyl-4',5'-dihydrooxazoline-N-oxyl 7, a potential spin probe for biomembranes is described. The title compound in improved yield could be obtained by a direct Grignard reaction on the oxaziridine 4. This effected a one-step reduction in the overall synthetic sequence. The methodology of the Grignard reaction on the oxaziridine to yield the nitroxide is reported for the first time. In dilute solutions, the isotropic ESR parameters for 7 have been measured.
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Publisher |
PERGAMON-ELSEVIER SCIENCE LTD
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Date |
2011-08-26T19:49:36Z
2011-12-26T12:57:35Z 2011-12-27T05:43:46Z 2011-08-26T19:49:36Z 2011-12-26T12:57:35Z 2011-12-27T05:43:46Z 1992 |
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Type |
Article
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Identifier |
TETRAHEDRON, 48(1), 133-148
0040-4020 http://dx.doi.org/10.1016/S0040-4020(01)80586-X http://dspace.library.iitb.ac.in/xmlui/handle/10054/11419 http://hdl.handle.net/10054/11419 |
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Language |
en
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