DIVERSITY-ORIENTED APPROACH TO 1,2,3,4-TETRAHYDROISOQUINOLINE-3-CARBOXYLIC ACID (TIC) DERIVATIVES USING DIETHYL ACETAMIDOMALONATE AS A GLYCINE EQUIVALENT : FURTHER EXPANSION BY SUZUKI-MIYAURA CROSS-COUPLING REACTION
DSpace at IIT Bombay
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Title |
DIVERSITY-ORIENTED APPROACH TO 1,2,3,4-TETRAHYDROISOQUINOLINE-3-CARBOXYLIC ACID (TIC) DERIVATIVES USING DIETHYL ACETAMIDOMALONATE AS A GLYCINE EQUIVALENT : FURTHER EXPANSION BY SUZUKI-MIYAURA CROSS-COUPLING REACTION
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Creator |
KOTHA, S
MISRA, S KRISHNA, NG DEVUNURI, N HOPF, H KEECHERIKUNNEL, A |
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Subject |
constrained phenylalanine derivatives
ring-closing metathesis diels-alder reaction synthetic approach strategic combination 2+2+2 cycloaddition enyne metathesis amino-acids chemistry rongalite unusual amino acid building block approach suzuki coupling reaction boronic acid |
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Description |
Synthesis of diverse 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Tic) derivatives and its higher analogues are reported using diethyl acetamidomalonate as a glycine equivalent. In addition, various substituted Tic derivatives are assembled by application of Suzuki-Miyaura cross-coupling reaction as a key step.
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Publisher |
PERGAMON-ELSEVIER SCIENCE LTD
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Date |
2011-08-24T02:56:38Z
2011-12-26T12:56:42Z 2011-12-27T05:45:51Z 2011-08-24T02:56:38Z 2011-12-26T12:56:42Z 2011-12-27T05:45:51Z 2010 |
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Type |
Article
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Identifier |
HETEROCYCLES, 80(2), 847-854
0385-5414 http://dx.doi.org/10.3987/COM-09-S(S)103 http://dspace.library.iitb.ac.in/xmlui/handle/10054/10734 http://hdl.handle.net/10054/10734 |
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Language |
en
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