Rauhut-Currier type homo- and heterocouplings involving nitroalkenes and nitrodienes
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Title |
Rauhut-Currier type homo- and heterocouplings involving nitroalkenes and nitrodienes
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Creator |
SHANBHAG, P
NAREDDY, PR DADWAL, M MOBIN, SM NAMBOOTHIRI, INN |
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Subject |
baylis-hillman reaction
pauson-khand reaction alpha,beta-unsaturated nitro-compounds dabco-catalyzed dimerization conjugated nitroalkenes anticancer activity michael cycloisomerization activated olefins acrylic compounds esters |
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Description |
Reaction of nitroalkenes or nitrodienes with methyl vinyl ketone (MVK) or acrylate in the presence of the imidazole-LiCl catalyst system provides Rauhut-Currier (vinylogous Morita-Baylis-Hillman) adducts in moderate yield. Under similar conditions (imidazole-hydroquinone), nitroalkenes and nitrodienes undergo self-dimerization to afford the Rauhut-Currier adducts in varying yields. An alternative self-dimerization-nitro group elimination pathway in the presence tricyclohexylphosphine was observed with heteroaromatic nitroalkenes. A synthetically useful one-pot two step transformation of Rauhut-Currier adducts of nitroalkenes with MVK to 2,3-disubstituted cyclopentenones is also described.
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Publisher |
ROYAL SOC CHEMISTRY
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Date |
2011-08-28T16:13:54Z
2011-12-26T12:58:06Z 2011-12-27T05:47:27Z 2011-08-28T16:13:54Z 2011-12-26T12:58:06Z 2011-12-27T05:47:27Z 2010 |
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Type |
Article
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Identifier |
ORGANIC & BIOMOLECULAR CHEMISTRY, 8(21), 4867-4873
1477-0520 http://dx.doi.org/10.1039/c0ob00062k http://dspace.library.iitb.ac.in/xmlui/handle/10054/11784 http://hdl.handle.net/10054/11784 |
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Language |
en
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