Stereoselective synthesis of (-)-1-epi-ventiloquinone L and (+)-ventiloquinone L, the monomeric unit of cardinalin 3
DSpace at IIT Bombay
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Title |
Stereoselective synthesis of (-)-1-epi-ventiloquinone L and (+)-ventiloquinone L, the monomeric unit of cardinalin 3
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Creator |
FERNANDES, RA
INGLE, AB CHAVAN, VP |
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Subject |
CHROMIUM-CARBENE COMPLEXES
DERMOCYBE CARDINALIS ALKYNE CYCLOADDITION (+)-NOCARDIONE B FORMAL SYNTHESIS VENTILOQUINONE-L (+)-ALLO-ELEUTHERIN (+)-ELEUTHERIN ANTIBIOTICS PIGMENTS |
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Description |
A stereoselective synthesis of (-)-1-epi-ventiloquinone L and (+)-ventiloquinone L, the monomeric unit of cardinalin 3 has been described. The synthesis is completed in 7 steps with 10.5% and 13% overall yields for (-)-1-epi-ventiloquinone L and (+)-ventiloquinone L respectively. The key steps involve Dotz benzannulation of carbene 5 with alkyne 6 to give a substituted naphthalene moiety and oxa-Pictet-Spengler reaction to install the 1,3-dimethylpyran moiety.
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Publisher |
ROYAL SOC CHEMISTRY
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Date |
2014-10-16T14:04:49Z
2014-10-16T14:04:49Z 2012 |
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Type |
Article
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Identifier |
ORGANIC & BIOMOLECULAR CHEMISTRY, 10(22)4462-4466
http://dx.doi.org/10.1039/c2ob25453k http://dspace.library.iitb.ac.in/jspui/handle/100/15738 |
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Language |
en
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