Enhancing Cubosome Functionality by Coating with a Single Layer of Poly-epsilon-lysine
DSpace at IIT Bombay
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Title |
Enhancing Cubosome Functionality by Coating with a Single Layer of Poly-epsilon-lysine
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Creator |
DESHPANDE, S
VENUGOPAL, E RAMAGIRI, S BELLARE, JR KUMARASWAMY, G SINGH, N |
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Subject |
bioconjugation
cubosomes drug delivery vehicle dual loading theranostics LIQUID-CRYSTALLINE DISPERSIONS DRUG-DELIVERY-SYSTEM IN-VITRO SUBMICRON PARTICLES NANOPARTICLES PHASES WATER VIVO CYTOTOXICITY EFFICIENCY |
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Description |
We report the preparation and characterization of monoolein cubosomes that can be easily surface modified through adsorption of a single layer of cationic poly-epsilon-lysine. Poly-epsilon-lysine coated cubosomes show remarkable stability in serum solution, are nontoxic and, are readily internalized by HeLa cells. The poly-epsilon-lysine coating provides chemical handles for further bioconjugation of the cubosome surface. We also demonstrate that the initial release rate of a hydrophilic drug, Naproxen sodium, from the cubosomes is retarded with just a single layer of polymer. Interestingly, cubosomes loaded with Naproxen sodium, recently shown to have anticancer properties, cause more apoptosis in HeLa cells when compared to free unencapsulated drug.
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Publisher |
AMER CHEMICAL SOC
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Date |
2014-12-29T05:33:43Z
2014-12-29T05:33:43Z 2014 |
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Type |
Article
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Identifier |
ACS APPLIED MATERIALS & INTERFACES, 6(19)17126-17133
1944-8244 http://dx.doi.org/10.1021/am5047872 http://dspace.library.iitb.ac.in/jspui/handle/100/17204 |
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Language |
English
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