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Synthesis of conformationally constrained alpha-amino acid derivatives containing bicyclo[2.2.2] unit via the Diels-Alder and Suzuki-Miyaura cross-coupling reactions as key steps

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Title Synthesis of conformationally constrained alpha-amino acid derivatives containing bicyclo[2.2.2] unit via the Diels-Alder and Suzuki-Miyaura cross-coupling reactions as key steps
 
Creator KOTHA, S
MESHRAM, M
MUTHUSAMY, G
 
Subject 9-SUBSTITUTED ANTHRACENES
PALLADIUM CATALYSTS
2-ACETAMIDOACRYLATE
BROMINATION
METATHESIS
TRIBROMIDE
DIVERSITY
PEPTIDES
HALIDES
Bicyclic alpha-amino acid derivatives
glycine equivalent
anthracene derivatives
Diels-Alder reaction
Suzuki-Miyaura cross-coupling reaction
Buchwald ligand
 
Description A simple route to synthesize conformationally constrained a-amino acid (AAA) derivatives containing bicyclo[2.2.2]octane ring-system has been devised. Diels-Alder reaction is chosen to assemble highly constrained AAA derivatives and the scope of the methodology is further expanded by Suzuki-Miyaura cross-coupling reaction with various boronic acids.
 
Publisher COUNCIL SCIENTIFIC & INDUSTRIAL RES
 
Date 2016-01-15T10:58:23Z
2016-01-15T10:58:23Z
2015
 
Type Article
 
Identifier INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 54(4)505-513
0376-4699
0019-5103
http://dspace.library.iitb.ac.in/jspui/handle/100/18406
 
Language en