QSAR based model for discriminating EGFR inhibitors and non-inhibitors using Random forest.
DIR@IMTECH: CSIR-Institute of Microbial Technology
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Title |
QSAR based model for discriminating EGFR inhibitors and non-inhibitors using Random forest.
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Creator |
Singh, Harinder
Singh, Sandeep Singla, Deepak Agarwal, Subhash M Raghava, G.P.S. |
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Subject |
QR Microbiology
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Description |
Epidermal Growth Factor Receptor (EGFR) is a well-characterized cancer drug target. In the past, several QSAR models have been developed for predicting inhibition activity of molecules against EGFR. These models are useful to a limited set of molecules for a particular class like quinazoline-derivatives. In this study, an attempt has been made to develop prediction models on a large set of molecules (~3500 molecules) that include diverse scaffolds like quinazoline, pyrimidine, quinoline and indole.
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Publisher |
BioMedCentral
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Date |
2015
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Type |
Article
PeerReviewed |
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Format |
application/pdf
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Identifier |
http://crdd.osdd.net/open/1638/1/GPSR%202015%20prot%20str%20functio%20...24783.pdf
Singh, Harinder and Singh, Sandeep and Singla, Deepak and Agarwal, Subhash M and Raghava, G.P.S. (2015) QSAR based model for discriminating EGFR inhibitors and non-inhibitors using Random forest. Biology direct, 10. p. 10. ISSN 1745-6150 |
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Relation |
http://www.biologydirect.com/content/10/1/10
http://crdd.osdd.net/open/1638/ |
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