C-Glycosylated flavonoids from black gram husk: Protection againstDNA and erythrocytes from oxidative damage and their cytotoxiceffect on HeLa cells.
IR@CSIR-CFTRI
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Relation |
http://ir.cftri.com/13260/
http://dx.doi.org/10.1016/j.toxrep.2016.08.006 |
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Title |
C-Glycosylated flavonoids from black gram husk: Protection againstDNA and erythrocytes from oxidative damage and their cytotoxiceffect on HeLa cells.
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Creator |
Girish, T. K.
Anil Kumar, K. Prasada Rao, U. J. S. |
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Subject |
18 Flavonoid Chemistry
07 Waste utilization 22 Legumes-Pulses |
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Description |
tC-Glycosyl flavones are present in different plant tissues and they exhibit health benefits. In the presentstudy, it was found that C-glycosyl flavones are distributed in different milled fractions of black gram andamong these fractions, husk had the highest content of C-glycosyl flavones. Two C-glycosyl flavones fromblack gram husk were extracted and purified by preparative high-performance liquid chromatography(HPLC) column. The purity of each compound was assessed by analytical C18 column. The structure of eachcompound was confirmed by LC–MS/MS, NMR. The molecular mass of these compounds were found to be[M−H]−, m/z 431.36 and [M−H]−, m/z 431.35 and were identified as vitexin and isovitexin, respectively.Content of vitexin and isovitexin in aqueous ethanol extract was found to be 76 and 65 mg/g of extract,respectively. These C-glycosyl flavones protected DNA and erythrocytes from oxidative damage. The IC50values for vitexin, isovitexin and quercetin for hemolysis were 6, 5.7 and 2.37 �g, respectively. Thesecompounds also triggered the process of apoptosis in HeLa cells by downregulating Bcl-2 level with thesimultaneous upregulation of Bax and caspase-3 protein expression. Thus, C-glycosyl flavones from blackgram husk protected DNA and erythrocytes from oxidative damage and exhibited anticancer activity.
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Date |
2016
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Type |
Article
PeerReviewed |
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Format |
pdf
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Language |
en
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Identifier |
http://ir.cftri.com/13260/1/Toxicology%20Reports%203%20%282016%29%20652%E2%80%93663.pdf
Girish, T. K. and Anil Kumar, K. and Prasada Rao, U. J. S. (2016) C-Glycosylated flavonoids from black gram husk: Protection againstDNA and erythrocytes from oxidative damage and their cytotoxiceffect on HeLa cells. Toxicology Reports, 3. pp. 652-663. |
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