Water-Soluble Tripeptide A� (9-11) Forms Amyloid-Like Fibrils and Exhibits Neurotoxicity
EPrints@IICB
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Title |
Water-Soluble Tripeptide A� (9-11) Forms Amyloid-Like Fibrils and Exhibits Neurotoxicity
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Creator |
Naskar, Jishu
Drew, Michael G B Deb, Ishani Das, Sumantra Banerjee, Arindam |
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Subject |
Chemistry
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Description |
The aggregation of normally soluble proteins into wellordered amyloid fibrils is associated with a number of diseases including Alzheimer’s disease, Parkinson’s disease, type II diabetes, prion-related diseases, and others.1 Among these diseases, Alzheimer’s disease (AD) is the most prevalent and progressive neurodegenerative disease associated with deposition of �-sheet-rich protein aggregates in specific regions of the human brain as amyloid fibrils,2 which consist mainly of amyloid peptides like A�(1-40) and A�(1- 42).3 A� peptides are generated from highly regulated and sequential cleavage of the amyloid precursor protein (APP) by proteases designated as �- and γ-secretases and are readily detected in human CSF4 as a range of isoforms between 38 and 43 amino acids in length. They normally exist as soluble random coils. However, in a diseased condition they misfold and form self-assembled oligomers which further selfassociate to form amyloid fibrils.5 The molecular structure of full-length A� fibrils is still not completely clear because of the difficulty of growing good quality crystals that can diffract well enough to obtain crystal structures. |
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Date |
2008
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Type |
Article
PeerReviewed |
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Format |
application/pdf
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Identifier |
http://www.eprints.iicb.res.in/189/1/ORGANIC_LETTERS%2C_10(_13)%2C_2625%2D2628%2C2008[52].pdf
Naskar, Jishu and Drew, Michael G B and Deb, Ishani and Das, Sumantra and Banerjee, Arindam (2008) Water-Soluble Tripeptide A� (9-11) Forms Amyloid-Like Fibrils and Exhibits Neurotoxicity. Organic Letters, 10 (13). pp. 2625-2528. |
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Relation |
http://dx.doi.org/10.1021/ol8007217
http://www.eprints.iicb.res.in/189/ |
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