Structural Analysis of Factor IX Protein Variants to Predict Functional Aberration Causing Haemophilia B
EPrints@IICB
View Archive InfoField | Value | |
Title |
Structural Analysis of Factor IX Protein Variants to Predict Functional Aberration Causing Haemophilia B |
|
Creator |
Mukherjee, S
Saha, A Biswas, P Mandal, C Ray, Kunal |
|
Subject |
Molecular & Human Genetics
|
|
Description |
Factor IX (FIX) is a vitamin K-dependent serine protease precursor that upon activation plays a crucial role in blood coagulation [1]. A lack of its coagulant activity results in haemophilia B, a bleeding disorder affecting nearly 30 000 male births worldwide. Human FIX is synthesized in the liver as a precursor molecule containing 461 amino acids, of which the first 46 residues are removed. During biosynthesis, the protein undergoes several post posttranslational modifications, which include c-carboxylation and hydroxylation. The resulting mature protein containing 415 amino acids is a zymogen of serine protease. Upon initiation of blood coagulation, either FVIIa or FXIa converts FIX to its active form FIXa by proteolysis. During this process, the activation peptide (residue 146–180) is cleaved off resulting in a two-chain molecule comprising of covalently linked light and heavy chains, which are organized into several distinct domains: an aminoterminal c-carboxyglutamic acid (Gla) domain (residues 1–40), a short hydrophobic segment (residues 41–46), two epidermal growth factor (EGF)-like domains [EGF1 residues (47–84) and EGF2 residues (85–127)] and a carboxyl-terminal serine protease domain. |
|
Date |
2008
|
|
Type |
Article
PeerReviewed |
|
Format |
application/pdf
|
|
Identifier |
http://www.eprints.iicb.res.in/296/1/HAEMOPHILIA%2C14(_5)%2C1076%2D1081%2C2008[41].pdf
Mukherjee, S and Saha, A and Biswas, P and Mandal, C and Ray, Kunal (2008) Structural Analysis of Factor IX Protein Variants to Predict Functional Aberration Causing Haemophilia B. Haemophilia, 14 (5). pp. 1076-1081. |
|
Relation |
http://dx.doi.org/10.1111/j.1365-2516.2008.01788.x
http://www.eprints.iicb.res.in/296/ |
|