Synthesis of Chiral Benzoxa(thia)zepine and Pyridoxazepine Derivatives Using Palladium-Catalyzed Intramolecular Aryl Amination Reaction.
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Title |
Synthesis of Chiral Benzoxa(thia)zepine and Pyridoxazepine Derivatives Using Palladium-Catalyzed Intramolecular Aryl Amination Reaction.
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Creator |
Das Adhikary, Nirmal
Chattopadhyay, Partha |
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Subject |
Chemistry
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Description |
A palladium-catalyzed method employing different bulky biaryl phosphanes as ligands has been developed for the intramolecular amination of aryl bromides and iodides. A variety of aryl halide substrates have been aminated through the intramolecular pathway in good yield using different sugar-derived amines to give furo-benzoxa(thia)zepine and pyridoxazepine derivatives. The method is capable of furnishing chiral, enantiopure benzoxa(thia)zepines and pyridoxazepines of significant biological importance. |
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Publisher |
John Wiley & Sons
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Date |
2011
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Type |
Article
PeerReviewed |
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Format |
application/pdf
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Identifier |
http://www.eprints.iicb.res.in/1258/1/EUROPEAN_JOURNAL_OF_ORGANIC_CHEMISTRY__(_36)_7346%2D7354;2011[5].pdf
Das Adhikary, Nirmal and Chattopadhyay, Partha (2011) Synthesis of Chiral Benzoxa(thia)zepine and Pyridoxazepine Derivatives Using Palladium-Catalyzed Intramolecular Aryl Amination Reaction. European Journal of Organic Chemistry, 36. 7346-7354 . ISSN 1434-193X |
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Relation |
http://dx.doi.org/10.1002/ejoc.201101174
http://www.eprints.iicb.res.in/1258/ |
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