Efficient Synthesis of Imidazole-Fused Benzodiazepines Using Palladium- Catalyzed Intramolecular C–N Bond Formation Reaction
EPrints@IICB
View Archive InfoField | Value | |
Title |
Efficient Synthesis of Imidazole-Fused Benzodiazepines Using Palladium- Catalyzed Intramolecular C–N Bond Formation Reaction |
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Creator |
Maitra, Sudipta
Darira, Heena Chattopadhyay, Partha |
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Subject |
Chemistry
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Description |
An efficient three-step synthetic route to imidazolefused benzodiazepines from imidazole-2-carbaldehyde is described. Application of intramolecular Buchwald–Hartwig cycloamination reaction in the final step is shown to be a convenient method for the synthesis of fused seven-membered diazacycles. The reactions proceeded smoothly with both aliphatic and aromatic amines. |
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Date |
2013
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Type |
Article
PeerReviewed |
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Format |
application/pdf
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Identifier |
http://www.eprints.iicb.res.in/1823/1/SYNTHESIS%2DSTUTTGART___45(_1)_85%2D92;2013[17].pdf
Maitra, Sudipta and Darira, Heena and Chattopadhyay, Partha (2013) Efficient Synthesis of Imidazole-Fused Benzodiazepines Using Palladium- Catalyzed Intramolecular C–N Bond Formation Reaction. Synthesis, 45 (1). pp. 85-92. |
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Relation |
http://dx.doi.org/10.1055/s-0032-1316828
http://www.eprints.iicb.res.in/1823/ |
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