Synthesis of Polynuclear Heteroaromatics Mainly Based on Pyridine and Quinoline
EPrints@IICB
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Title |
Synthesis of Polynuclear Heteroaromatics Mainly Based on Pyridine and Quinoline
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Creator |
Paira, Rupankar
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Subject |
Chemistry
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Description |
The thesis embodies the results of studies on the “Synthesis of polynuclear heteroaromatics mainly based on pyridine and quinoline”. Quinoline and pyridine derivatives are a class of synthetic antibiotics with broad spectrum of antibacterial as well as anti-malarial activities. The fused pyridine and quinoline derivatives are also known to be effective in the treatment of autoimmune conditions (such as rhenumatoid arthritis) with their anti inflammatory effects. Among the numerous structurally diverse derivatives of pyridine and quinolines many show significant biological activity such as quinine, morphine, and multifloramine. Hence, it is not surprising that this structural motif is also an important component in many of today’s pharmaceuticals. Nevertheless, the diversity of pyridine and quinoline as well as their biological and pharmaceutical relevance is still motivating academic and industrial researchers to look for new and improved syntheses for quinoline derivatives. Clearly, a number of practical methods have been developed for the synthesis of pyridine and quinolines in the past century. More recently, especially transition metal catalysis has become a powerful tool for synthetic methodology but chemical and biological research has now presented a great challenge to synthesize and optimise highly efficient and cost-effective synthetic routes to some unique and novel biologically active substances. |
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Date |
2012
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Type |
Thesis
NonPeerReviewed |
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Format |
application/pdf
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Identifier |
http://www.eprints.iicb.res.in/1844/1/Rupankar_Paira_%2D_Thesis.pdf
Paira, Rupankar (2012) Synthesis of Polynuclear Heteroaromatics Mainly Based on Pyridine and Quinoline. PhD thesis, Jadavpur University. |
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Relation |
http://www.eprints.iicb.res.in/1844/
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