<strong>One-pot synthesis of coumarin derivatives via microwave assisted Pechmann reaction and biological activity of substituted coumarin derivatives</strong>
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Title Statement |
<strong>One-pot synthesis of coumarin derivatives via microwave assisted Pechmann reaction and biological activity of substituted coumarin derivatives</strong> |
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Added Entry - Uncontrolled Name |
Sharma, Dipak ; Maharaja Ranjit Singh College of Professional Sciences Indore (M.P.) monga, paramjeet ; Suresh Gyan Vihar University jaipur bhasin, Sheetal ; Maharaja Ranjit Singh College of Professional Sciences Indore (M.P.) Dubey, Arti ; Viva College, Virar, M.S. Nagar, Hariom ; Suresh Gyan Vihar University, Jaipur, Rajasthan, India |
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Uncontrolled Index Term |
Antimicrobial; Antifungal; Coumarins; One-pot Microwave irradiation; Oxalic acid;Pechmann condensation |
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Summary, etc. |
Pechmann reaction is mainly used for the synthesis of substituted coumarins as it can be executed with straight forward primary resources and gives coumarin derivatives with excellent yields. In the present work coumarin derivatives have been synthesized by condensation of β-ketoesters and substituted phenols under microwave irradiation in solvent free condition in which oxalic acid is used as catalyst. Oxalic acid is found to be a potential environment friendly catalyst for synthesis of coumarins. The new method of synthesis described here offers a number of advantages of being convenient, safe, gentle, shorter reaction time, high yield, and cleanness as compared to the conventional methods. The synthesized compounds have been systematically characterized by IR and MS analyses. All products are examined for antimicrobial activity against the Gram positive (<em>Staphylococcus aureus</em> and <em>Bacillus subtilis</em>) and Gram negative (<em>Escherichia coli</em> and<em> Salmonella typhi</em>) bacteria and antifungal activity against two fungal species (<em>Aspergillus sp. </em>and<em> Fusarium graminearum</em>). All the compounds inhibited the growth of bacteria as well as fungi. |
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Publication, Distribution, Etc. |
Indian Journal of Chemical Technology (IJCT) 2020-08-21 13:49:58 |
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Electronic Location and Access |
application/pdf http://op.niscair.res.in/index.php/IJCT/article/view/21023 |
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Data Source Entry |
Indian Journal of Chemical Technology (IJCT); ##issue.vol## 27, ##issue.no## 2 (2020): Indian Journal of Chemical Technology |
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Language Note |
en |
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Nonspecific Relationship Entry |
http://op.niscair.res.in/index.php/IJCT/article/download/21023/465465473 http://op.niscair.res.in/index.php/IJCT/article/download/21023/465465474 http://op.niscair.res.in/index.php/IJCT/article/download/21023/465465475 http://op.niscair.res.in/index.php/IJCT/article/download/21023/465465476 http://op.niscair.res.in/index.php/IJCT/article/download/21023/465465477 http://op.niscair.res.in/index.php/IJCT/article/download/21023/465465478 |
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