CT-DNA-binding and biological activity of mononuclear copper(II) complexes with imidazo-phenanthroline ligands
NOPR - NISCAIR Online Periodicals Repository
View Archive InfoField | Value | |
Title |
CT-DNA-binding and biological activity of mononuclear copper(II) complexes with imidazo-phenanthroline ligands
|
|
Creator |
Nagababu, Penumaka
Thulasiram, B Nagarkar, Jidnyasa Devi, C Shobha Paul, Perala Sudheer Reddy, Thatiparthi Byragi |
|
Subject |
Cu(II) complexes
DNA-binding Docking studies Anti-cancer activity |
|
Description |
37-44
Four imidazo-phenanthroline (IP) based ligands and its corresponding copper polypyridyl complexes have been prepared [Cu(L1-L4)2]2+ and characterized by various physicochemical techniques. Herein we are reporting the CT-DNA (calf-thymus DNA) binding & anti-cancer affinity of ligands (L1-L4) as well as complexes (C1-C4). The DNA binding affinity of synthesized C1-C4 has been carried out by using spectroscopic techniques like UV/visible, emission, molecular modeling and viscosity techniques. The obtained results are clearly indicating that all C1-C4 complexes bind to DNA via intercalative mode and they possess a significant cytotoxic effect toward selected cancer cell lines (MDA-MB-231, B16-F10, DU-145 and CHO-K1). |
|
Date |
2021-01-12T09:24:47Z
2021-01-12T09:24:47Z 2021-01 |
|
Type |
Article
|
|
Identifier |
0975-0975(Online); 0376-4710(Print)
http://nopr.niscair.res.in/handle/123456789/55939 |
|
Language |
en_US
|
|
Rights |
CC Attribution-Noncommercial-No Derivative Works 2.5 India
|
|
Publisher |
NISCAIR-CSIR, India
|
|
Source |
IJC-A Vol.60A(01) [January 2021]
|
|