Synthesis and biological evaluation of novel 3-aryl-4-methoxy N-alkyl maleimides
NOPR - NISCAIR Online Periodicals Repository
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Title |
Synthesis and biological evaluation of novel 3-aryl-4-methoxy N-alkyl maleimides
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Creator |
Gosavi, Kirankumar S
Mahale, Keshao A Patil, Nilesh S Patil, Sambhaji V |
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Subject |
Maleimide
Maleic anhydride MIC Antifungal Antibacterial |
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Description |
473-478
In the present investigation, a series of 3-aryl-4-methoxy N-alkyl maleimide 5a-l have been synthesized and screened for their antimicrobial activity against one Gram positive bacteria (S. aureus), one Gram negative bacteria (E. coli) and fungal strains (C. albicans, C. tropicalis, A. niger and A. clavatus). The structures of the compounds have been substantiated by their IR, NMR, mass and elemental analysis. The minimum inhibitory concentrations (MICs) of synthesized maleimides have been determined by broth microdilution method. Of the newly synthesized maleimides, compounds 5c, 5f, 5h, 5i, 5k and 5l registered significant activity against the tested microorganisms. |
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Date |
2021-03-03T04:48:40Z
2021-03-03T04:48:40Z 2021-03 |
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Type |
Article
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Identifier |
0975-0983(Online); 0376-4699(Print)
http://nopr.niscair.res.in/handle/123456789/56384 |
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Language |
en_US
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Rights |
CC Attribution-Noncommercial-No Derivative Works 2.5 India
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Publisher |
NISCAIR-CSIR, India
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Source |
IJC-B Vol.60B(03) [March 2021]
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