Synthesis of isomeric naphthofuranyl coumarins as anti-inflammatory and analgesic agents
NOPR - NISCAIR Online Periodicals Repository
View Archive InfoField | Value | |
Title |
Synthesis of isomeric naphthofuranyl coumarins as anti-inflammatory and analgesic agents
|
|
Creator |
Yaragatti, Naazneen
Khanapurmath, Netravati Kulkarni, Manohar V |
|
Subject |
Naphthofuranyl
coumarin anti-inflammatory analgesic activity angular/linear naphthofuranyl coumarins |
|
Description |
1007-1013
A two-step synthetic scheme has been employed for the synthesis of 4-naphtho [2, 1-b] furan-2-yl-chromen-2-ones/4-(3-alkoxy-naphtho-[2,3-b]furan-2-yl)-chromen-2-ones(angular/linear naphthofuranyl coumarins). The reactions have been monitored by TLC and structures of the intermediates and the target compounds have been ascertained by IR, NMR and mass spectral data. Both the isomeric naphthofuranyl coumarins have been found to exhibit anti-inflammatory activity comparable to asprin but when tested for analgesic activity, angularly fused naphthofuranyl coumarins show better activity comparable to asprin whereas linear naphthofuranyl coumarins are less active. |
|
Date |
2021-09-29T07:17:55Z
2021-09-29T07:17:55Z 2021-07 |
|
Type |
Article
|
|
Identifier |
0975-0983(Online); 0376-4699(Print)
http://nopr.niscair.res.in/handle/123456789/58177 |
|
Language |
en
|
|
Publisher |
NIScPR-CSIR, India
|
|
Source |
IJC-B Vol.60B(07) [July 2021]
|
|