<p>Synthesis of bis chalcones and transformation into bis heterocyclic compounds with expected antimicrobial activity</p><p> </p>
Online Publishing @ NISCAIR
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Title Statement |
<p>Synthesis of bis chalcones and transformation into bis heterocyclic compounds with expected antimicrobial activity</p><p> </p> |
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Added Entry - Uncontrolled Name |
ghoneim, amira atef Manoer, Afaf ; Chemistry Department, College of Science, Jouf University, PO Box 2014, Sakaka, Aljouf, Kingdom of Saudi Arabia Elbargisy, Rehab M; Department of Pharmaceutics, College of Pharmacy, Jouf University, Sakaka, Al Jouf, Kingdom of Saudi Arabia Department of Microbiology and Immunology, Faculty of Pharmacy, Mansoura University, Mansoura 35516, Egypt |
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Uncontrolled Index Term |
Synthesis, bis chalcones, heterocyclic, ethylcyanoacetate, cyanopyridine |
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Summary, etc. |
<p>One-pot synthesis of novel derivatives of bis-chalcones has been achieved by condensation of 1,4-diacetylbenzene with different aldehydes in basic media. The reaction of chalcone derivatives <strong>3a,b</strong> with thioglycolic acid gives compounds <strong>4a,b</strong>. This, when reacted with ethyl cyanoacetate in presence of ammonium acetate gives the corresponding cyanopyridine derivatives <strong>5a,b</strong>. Furthermore, bis-chalcone <strong>3a,b</strong> has been cyclized to pyrazole analogs by using 2,4-dinitrophenylhydrazine to give compounds <strong>7a,b </strong>in good yields. All products have been characterized by IR, <sup>1</sup>H and <sup>13</sup>C NMR, and elemental analysis. The newly synthesised compounds<em> </em>have been screened for anti-bacterial activity.</p><p> </p> |
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Publication, Distribution, Etc. |
Indian Journal of Chemistry -Section B (IJC-B) 2021-10-14 15:19:06 |
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Electronic Location and Access |
application/pdf http://op.niscair.res.in/index.php/IJCB/article/view/30343 |
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Data Source Entry |
Indian Journal of Chemistry -Section B (IJC-B); ##issue.vol## 60, ##issue.no## 9 (2021): Indian Journal of Chemistry- Section-B, (IJCB) |
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Language Note |
en |
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Terms Governing Use and Reproduction Note |
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