<p>Synthesis, spectral characterization and anti-diabetic activity evaluation of phosphoramidate derivatives</p>
Online Publishing @ NISCAIR
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dc |
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Title Statement |
<p>Synthesis, spectral characterization and anti-diabetic activity evaluation of phosphoramidate derivatives</p> |
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Added Entry - Uncontrolled Name |
Ravikumar, D ; Department of Chemistry, Bapatla Engineering College, Bapatla 522 101, India Subramanyam, Ch ; Department of Chemistry, Bapatla Engineering College, Bapatla 522 101, India Venkataramaiah, Ch ; Division of Molecular Biology, Department of Zoology, Sri Venkateswara University, Tirupati 517 502, India Rajendra, W ; Division of Molecular Biology, Department of Zoology, Sri Venkateswara University, Tirupati 517 502, India Rao, K Prasada; Department of Chemistry, Bapatla Engineering College, Bapatla 522 101, India |
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Uncontrolled Index Term |
Phosphoramidates, 4-chlorobenzene sulfonyl chloride, molecular docking studies, anti-diabetic activity |
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Summary, etc. |
<p style="text-align: justify;">In the present work, a series of new phosphoramidate derivatives have been conveniently synthesized by using 4-chlorobenzene-sulfonyl chloride as preliminary material <em>via</em> substituted sulfonamides as intermediates with high yields in a short period by conventional and microwave irradiation techniques. All the synthesized compound have been characterized by spectral and elemental analyses. An <em>in silico</em> molecular docking study has been performed to find potent anti-diabetic drugs. <em>In vitro</em> anti-diabetic activity of the title compounds have also been screened by standard α-amylase inhibition assay. Some of the tested compounds have been proven to possess promising activity when compared with reference drug.</p> |
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Publication, Distribution, Etc. |
Indian Journal of Chemistry (IJC) 2022-02-02 16:02:00 |
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Electronic Location and Access |
application/pdf application/pdf http://op.niscair.res.in/index.php/IJC/article/view/60061 |
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Data Source Entry |
Indian Journal of Chemistry (IJC); ##issue.vol## 61, ##issue.no## 1 (2022): Indian Journal of Chemistry-(IJC) |
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Language Note |
en |
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