Synthesis and antimicrobial activity of novel benzo[4', 5']-imidazo[1',2':1,2]pyrrolo[3,4-b]isoxazolo[4,5-e]pyridines
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Title |
Synthesis and antimicrobial activity of novel benzo[4', 5']-imidazo[1',2':1,2]pyrrolo[3,4-b]isoxazolo[4,5-e]pyridines
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Creator |
Prasoona, G
Kishore, B Brahmeshwari, G |
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Subject |
1-(Prop-2-yn-1-yl)-1H-benzo[d]imidazo-2-carbaldehydes
condensation intramolecular Povarov reaction benzo[4',5']imidazo[1',2':1,2]pyrrolo[3,4-b]isoxazolo[4,5-e] pyridines antimicrobial activity |
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Description |
174-183
Synthesis of novel benzo [4',5'] imidazo [1',2':1,2] pyrrolo [3,4-b] isoxazolo [4,5-e] pyridines 8 has been achieved by reaction of 1-(prop-2-yn-1-yl)-1H-benzo [d] imidazo-2-carbaldehydes 5 with 5-amino -3-methylisoxazole 6 in presence of InCl3 in CH3CN media, followed by reaction of imine 7 with BF3.Et2O in DCE at 80°C. The newly synthesized title compounds 8 have been evaluated for their in vitro antimicrobial activity. Compounds 8 exhibit potent antimicrobial activity compared to that of standard drugs. |
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Date |
2022-02-16T06:01:10Z
2022-02-16T06:01:10Z 2022-02 |
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Type |
Article
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Identifier |
2583-1321 (Online); 0019-5103 (Print)
http://nopr.niscair.res.in/handle/123456789/59191 |
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Language |
en
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Publisher |
NIScPR-CSIR, India
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Source |
IJC Vol.61(02) [February 2022]
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