Influence of Escherichia coli lipopolysaccharide induced fever on the plasma kinetics of pazufloxacin in buffalo calves
Indian Agricultural Research Journals
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Title |
Influence of Escherichia coli lipopolysaccharide induced fever on the plasma kinetics of pazufloxacin in buffalo calves
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Creator |
SHARMA, S K
ADITI, ADITI UL HAQ, SHAH AHSAN |
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Subject |
Buffalo calves
Pazufloxacin Dosage regimen Fever Pharmacokinetics |
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Description |
The pharmacokinetics of pazufloxacin was studied in healthy and febrile buffalo calves (5 mg/kg, IV). The fever was induced with Escherichia coli lipopolysaccharide. The drug concentration in plasma was detected by HPLC method. At 2.5 min the concentration of pazufloxacin in healthy and febrile animals were 17.8 0.6 µg/ml and 15.4±0.5 mg/ml, respectively and drug was detected up to 16 h. The distribution half-life of pazufloxacin increased from 0.09±0.01 h in healthy animals to 0.16±0.01 h in febrile animals. Drug distribution was altered by fever as febrile animals showed higher volume of distribution (1.35 0.09 L/ kg) higher than normal animal (1.03±0.06 L/kg). Total body clearances in healthy and febrile animals were 539.7±28.3 and 510.6±18.2 ml/kg/h, respectively. To maintain minimum therapeutic concentration of 0.1 µg/ml, a satisfactory dosage regimen of pazufloxacin in healthy and febrile buffalo calves would be 4.7 mg/kg and 4 mg/kg body weight, respectively, to be repeated at 12 h intervals.
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Publisher |
Indian Council of Agricultural Research
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Date |
2014-02-12
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Type |
info:eu-repo/semantics/article
info:eu-repo/semantics/publishedVersion |
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Format |
application/pdf
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Identifier |
https://epubs.icar.org.in/index.php/IJAnS/article/view/37836
10.56093/ijans.v84i2.37836 |
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Source |
The Indian Journal of Animal Sciences; Vol. 84 No. 2 (2014); 166–169
2394-3327 0367-8318 |
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Language |
eng
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Relation |
https://epubs.icar.org.in/index.php/IJAnS/article/view/37836/16968
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Rights |
Copyright (c) 2014 The Indian Journal of Animal Sciences
https://creativecommons.org/licenses/by-nc-sa/4.0 |
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