Efficient synthesis, molecular docking and biological evaluation of novel isatine linked spiroheterocycle through multi-component reaction
NOPR - NISCAIR Online Periodicals Repository
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Title |
Efficient synthesis, molecular docking and biological evaluation of novel isatine linked spiroheterocycle through multi-component reaction
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Creator |
Gamit, Kumar G
Patel, Navin B Chabhadiya, Bhadresh Kumar K Jauhari, Smita |
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Subject |
N-Mannich base
Isatine Gabbapentin-lactum Antibacterial activity Antifungal activity |
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Description |
400-406
In this work, twelve compounds have been newly synthesized by one pot N-Mannich base multicomponent reaction. The synthesized compounds have been characterized by using FT-IR, 1H and 13C NMR and mass spectrometry. The final compounds have been evaluated for their in vitro antibacterial and antifungal activity using agar-well diffusion method. The tested compounds show poor to good activity with inhibition zone value between 8 to 25 mm, when compared to reference Ciprofloxacin and Flocanazole. Among them compounds 6b, 6c, 6d and 6g show most promoting activity against E.coli, B. cereus, B. substilis, A. niger and R. nigricans. |
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Date |
2024-04-16T08:54:48Z
2024-04-16T08:54:48Z 2024-04 |
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Type |
Article
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Identifier |
2583-1321 (Online); 0019-5103 (Print)
http://nopr.niscpr.res.in/handle/123456789/63773 https://doi.org/10.56042/ijc.v63i4.7109 |
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Language |
en
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Publisher |
NIScPR-CSIR, India
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Source |
IJC Vol.63(04) [April 2024]
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