Computational investigation on the impact of point mutations on the N-terminal domain of SHANK3, indicating distinct synaptopathies in Autism spectrum disorder
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Title |
Computational investigation on the impact of point mutations on the N-terminal domain of SHANK3, indicating distinct synaptopathies in Autism spectrum disorder
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Creator |
Almaadani, Hiba Khalil
Mattaparthi, Venkata Satish Kumar |
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Subject |
ASD
Molecular dynamics simulation P141A and L270M mutations SPN-ARR domains |
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Description |
527-538
SHANK3 mutations are associated with a notable 1% of autism spectrum disorder (ASD). Due to the cost and time associated with experimental polymorphism studies, in silico investigations are deemed a rational precursor to elucidate the role of two mutations implicated in ASD, SHANK3 P141A and SHANK3 L270M. ASD is a complex neurological condition with diverse clinical manifestations, encompassing challenges in social interaction, communication, and repetitive behaviors. ASD is characterized by genetic heterogeneity, converging on a limited set of molecular pathways. Synaptopathies are one of the common neuronal processes associated with ASD, involving altered glutamatergic that may disrupt the excitatory and inhibitory equilibrium. SHANK3 is pivotal as a scaffold protein connecting glutamate receptors to the cytoskeleton, crucial for synaptic transmission within the post-synaptic density. We conducted a 200 ns molecular dynamics simulation to explore SHANK3 P141A and SHANK3 L270M functional and structural consequences on the SHANK3 protein. The P141A mutation significantly disrupted SHANK3 stabilization and caused a disturbance in intramolecular connections between SPN and ARR domains. The alteration affected the αCaMKII binding as one of the pivotal protein partners. On the contrary, the SHANK3 L270M mutation resulted in moderate stability conformation. The findings underscore the intricate dynamics of SHANK3 mutations and their potential relevance to the ASD. |
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Date |
2024-08-29T10:18:29Z
2024-08-29T10:18:29Z 2024-08 |
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Type |
Article
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Identifier |
0975-0959 (Online); 0301-1208 (Print)
http://nopr.niscpr.res.in/handle/123456789/64463 https://doi.org/10.56042/ijbb.v61i9.10442 |
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Language |
en
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Publisher |
NIScPR-CSIR,India
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Source |
IJBB Vol.61(09) [September 2024]
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