Platinum(II) complexes of S-benzyldithiocarbazate based Schiff base ligand: Green synthesis, characterization, cytotoxic and antioxidant assay
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Title |
Platinum(II) complexes of S-benzyldithiocarbazate based Schiff base ligand: Green synthesis, characterization, cytotoxic and antioxidant assay
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Creator |
Jain, Akshita
Bhatnagar, Shivansh Dave, Saurabh Fahmi, Nighat |
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Subject |
S-Benzyldithiocarbazate
Pt(II) complexes Cytotoxic activity Antioxidant activity |
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Description |
1121-1129
In the present work, benzyl-2-((5-methylthiophen-2-yl)methylene)hydrazine-1-carbothiolate ligand and its platinum(II) complexes have been prepared by conventional and microwave assisted methods. Structural elucidation of the ligand and its Pt(II) complexes have been performed by elemental analysis, conductance measurements, mass spectrometry, powder XRD, FT-IR and 1H NMR spectroscopic methods. On the basis of analytical and spectral data, a square planar geometry has been suggested for the metal complexes. Starting material (PtCl2), Ligand (LH), metal complexes [Pt(L)2] and [Pt(LH)2]Cl2 have been screened for in vitro cytotoxic and antioxidant activity. Cytotoxic activity has been performed by MTT[3-(4,5- dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide] assay against cervical cancer (HeLa) cell line and human breast adenocarcinoma (MCF-7) cell line. Cisplatin has been used as the standard drug. [Pt(LH)2]Cl2 complex have shown better cytotoxicity in comparison to ligand and other complex with IC50 values of 72.76 μM and 59.93 μM against HeLa and MCF-7 respectively. The antioxidant activity has been measured in terms of radical scavenging ability using the stable radical DPPH. Ascorbic acid has been used as positive control and methanol is used as negative control. The ligand shows excellent antioxidant activity with 70.82% DPPH inhibition. |
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Date |
2024-11-20T04:59:16Z
2024-11-20T04:59:16Z 2024-11 |
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Type |
Article
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Identifier |
2583-1321 (Online); 0019-5103 (Print)
http://nopr.niscpr.res.in/handle/123456789/64887 https://doi.org/10.56042/ijc.v63i11.12888 |
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Language |
en
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Publisher |
NIScPR-CSIR, India
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Source |
IJC Vol.63(11) [November 2024]
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